Reduced treatment frequencies with bumped kinase inhibitor 1369 are effective against porcine cystoisosporosis
Publication date: Available online 21 August 2020Source: International Journal for Parasitology: Drugs and Drug ResistanceAuthor(s): Aruna Shrestha, Bärbel Ruttkowski, Patricia Greber, Grant R. Whitman, Matthew A. Hulverson, Ryan Choi, Samantha A. Michaels, Kayode K. Ojo, Wesley C. Van Voorhis, Anja Joachim (Source: International Journal for Parasitology: Drugs and Drug Resistance)
Source: International Journal for Parasitology: Drugs and Drug Resistance - August 22, 2020 Category: Parasitology Source Type: research

Quantitative benzimidazole resistance and fitness effects of parasitic nematode beta-tubulin alleles
Publication date: Available online 20 August 2020Source: International Journal for Parasitology: Drugs and Drug ResistanceAuthor(s): Clayton M. Dilks, Steffen R. Hahnel, Qicong Sheng, Lijiang Long, Patrick T. McGrath, Erik C. Andersen (Source: International Journal for Parasitology: Drugs and Drug Resistance)
Source: International Journal for Parasitology: Drugs and Drug Resistance - August 21, 2020 Category: Parasitology Source Type: research

RNA interference dynamics in juvenile Fasciola hepatica are altered during in vitro growth and development
Publication date: Available online 19 August 2020Source: International Journal for Parasitology: Drugs and Drug ResistanceAuthor(s): Paul McCusker, Wasim Hussain, Paul McVeigh, Erin McCammick, Nathan G. Clarke, Emily Robb, Fiona M. McKay, Peter M. Brophy, David J. Timson, Angela Mousley, Nikki J. Marks, Aaron G. Maule (Source: International Journal for Parasitology: Drugs and Drug Resistance)
Source: International Journal for Parasitology: Drugs and Drug Resistance - August 21, 2020 Category: Parasitology Source Type: research

Repurposing bioenergetic modulators against protozoan parasites responsible for tropical diseases
Publication date: December 2020Source: International Journal for Parasitology: Drugs and Drug Resistance, Volume 14Author(s): Alba Martínez-Flórez, Melina Galizzi, Luis Izquierdo, Juan M. Bustamante, Ana Rodriguez, Fernando Rodriguez, Alhelí Rodríguez-Cortés, Jordi Alberola (Source: International Journal for Parasitology: Drugs and Drug Resistance)
Source: International Journal for Parasitology: Drugs and Drug Resistance - August 21, 2020 Category: Parasitology Source Type: research

Antileishmanial activity of a new chloroquine analog in an animal model of Leishmania panamensis infection
Publication date: Available online 15 August 2020Source: International Journal for Parasitology: Drugs and Drug ResistanceAuthor(s): Lizzi Herrera, Alejandro Llanes, Jennifer Álvarez, Kissy Degracia, Carlos M. Restrepo, Rene Rivera, David E. Stephens, Hang T. Dang, Oleg V. Larionov, Ricardo Lleonart, Patricia L. Fernandez (Source: International Journal for Parasitology: Drugs and Drug Resistance)
Source: International Journal for Parasitology: Drugs and Drug Resistance - August 15, 2020 Category: Parasitology Source Type: research

Activity of paromomycin against Leishmania amazonensis: Direct correlation between susceptibility in vitro and the treatment outcome in vivo
Publication date: Available online 15 August 2020Source: International Journal for Parasitology: Drugs and Drug ResistanceAuthor(s): Elizabeth M. Coser, Bianca A. Ferreira, Nilson Branco, Edite H. Yamashiro-Kanashiro, José Angelo L. Lindoso, Adriano C. Coelho (Source: International Journal for Parasitology: Drugs and Drug Resistance)
Source: International Journal for Parasitology: Drugs and Drug Resistance - August 15, 2020 Category: Parasitology Source Type: research

Where are all the anthelmintics? Challenges and opportunities on the path to new anthelmintics
Publication date: Available online 29 July 2020Source: International Journal for Parasitology: Drugs and Drug ResistanceAuthor(s): Samantha A. Nixon, Claudia Welz, Debra Woods, Livio Costa-Junior, Mostafa Zamanian, Richard Martin (Source: International Journal for Parasitology: Drugs and Drug Resistance)
Source: International Journal for Parasitology: Drugs and Drug Resistance - July 31, 2020 Category: Parasitology Source Type: research

A conserved coccidian gene is involved in Toxoplasma sensitivity to the anti-apicomplexan compound, tartrolon E
Publication date: Available online 25 July 2020Source: International Journal for Parasitology: Drugs and Drug ResistanceAuthor(s): Gregory D. Bowden, Patricia M. Reis, Maxwell B. Rogers, Rachel M. Bone Relat, Kelly A. Brayton, Sarah K. Wilson, Bruno Martorelli Di Genova, Laura J. Knoll, Felix J. Nepveux V, Albert K. Tai, Timothy R. Ramadhar, Jon Clardy, Roberta M. O'Connor (Source: International Journal for Parasitology: Drugs and Drug Resistance)
Source: International Journal for Parasitology: Drugs and Drug Resistance - July 26, 2020 Category: Parasitology Source Type: research

Energy blackout against glycolytic parasites
Publication date: Available online 22 July 2020Source: International Journal for Parasitology: Drugs and Drug ResistanceAuthor(s): Alba Martínez-Flórez, Melina Galizzi, Luis Izquierdo, Juan M. Bustamante, Fernando Rodriguez, Alhelí Rodríguez-Cortés, Jordi Alberola (Source: International Journal for Parasitology: Drugs and Drug Resistance)
Source: International Journal for Parasitology: Drugs and Drug Resistance - July 24, 2020 Category: Parasitology Source Type: research

Drug repurposing applied: Activity of the anti-malarial mefloquine against Echinococcus multilocularis
Publication date: Available online 2 July 2020Source: International Journal for Parasitology: Drugs and Drug ResistanceAuthor(s): Britta Lundström-Stadelmann, Reto Rufener, Andrew Hemphill (Source: International Journal for Parasitology: Drugs and Drug Resistance)
Source: International Journal for Parasitology: Drugs and Drug Resistance - July 3, 2020 Category: Parasitology Source Type: research

Mode of action of a formulation containing hydrazones and saponins against leishmania spp. Role in mitochondria, proteases and reinfection process
Publication date: Available online 26 June 2020Source: International Journal for Parasitology: Drugs and Drug ResistanceAuthor(s): Yulieth A. Upegui Zapata, Fernando Echeverri, Winston Quiñones, Fernando Torres, Montserrat Nacher, Luis I. Rivas, Camila dos Santos Meira, Lashitew Gedamu, Gustavo Escobar, Rosendo Archbold, Iván D. Vélez, Sara M. Robledo (Source: International Journal for Parasitology: Drugs and Drug Resistance)
Source: International Journal for Parasitology: Drugs and Drug Resistance - June 28, 2020 Category: Parasitology Source Type: research

Repurposing the open access malaria box reveals compounds with activity against Tritrichomonas foetus trophozoites
Publication date: Available online 17 June 2020Source: International Journal for Parasitology: Drugs and Drug ResistanceAuthor(s): Katy A. Martin, Jeba R.J. Jesudoss Chelladurai, Christopher Bader, Elizabeth Carreiro, Katelyn Long, Kylie Thompson, Matthew T. Brewer (Source: International Journal for Parasitology: Drugs and Drug Resistance)
Source: International Journal for Parasitology: Drugs and Drug Resistance - June 18, 2020 Category: Parasitology Source Type: research

Novel structural CYP51 mutation in Trypanosoma cruzi associated with multidrug resistance to CYP51 inhibitors and reduced infectivity
Publication date: Available online 13 June 2020Source: International Journal for Parasitology: Drugs and Drug ResistanceAuthor(s): Caio H. Franco, David C. Warhurst, Tapan Bhattacharyya, Ho Y.A. Au, Hai Le, Miriam A. Giardini, Bruno S. Pascoalino, Ana Claudia Torrecilhas, Lavinia M.D. Romera, Rafael Pedro Madeira, Sergio Schenkman, Lucio H. Freitas-Junior, Eric Chatelain, Michael A. Miles, Carolina B. Moraes (Source: International Journal for Parasitology: Drugs and Drug Resistance)
Source: International Journal for Parasitology: Drugs and Drug Resistance - June 14, 2020 Category: Parasitology Source Type: research

In vitro activity of Camellia sinensis (green tea) against trophozoites and cysts of Acanthamoeba castellanii
Publication date: Available online 2 June 2020Source: International Journal for Parasitology: Drugs and Drug ResistanceAuthor(s): Lenu B. Fakae, Carl W. Stevenson, Xing-Quan Zhu, Hany M. Elsheikha (Source: International Journal for Parasitology: Drugs and Drug Resistance)
Source: International Journal for Parasitology: Drugs and Drug Resistance - June 3, 2020 Category: Parasitology Source Type: research

Identification of annotated bioactive molecules that impair motility of the blood fluke Schistosoma mansoni
Publication date: Available online 1 June 2020Source: International Journal for Parasitology: Drugs and Drug ResistanceAuthor(s): Thomas B. Duguet, Anastasia Glebov, Asimah Hussain, Shashank Kulkarni, Igor Mochalkin, Timothy G. Geary, Mohammed Rashid, Thomas Spangenberg, Paula Ribeiro (Source: International Journal for Parasitology: Drugs and Drug Resistance)
Source: International Journal for Parasitology: Drugs and Drug Resistance - June 1, 2020 Category: Parasitology Source Type: research