Design, synthesis, and molecular modeling of heterocyclic bioisostere as potent PDE4 inhibitors
Archiv der Pharmazie, EarlyView. (Source: Archiv der Pharmazie)
Source: Archiv der Pharmazie - March 24, 2018 Category: Drugs & Pharmacology Source Type: research
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Archiv der Pharmazie, Ahead of Print. (Source: Archiv der Pharmazie)
Source: Archiv der Pharmazie - March 24, 2018 Category: Drugs & Pharmacology Source Type: research
Design, synthesis, and neuroprotective effects of dual ‐brain targeting naproxen prodrug
Archiv der Pharmazie, EarlyView. (Source: Archiv der Pharmazie)
Source: Archiv der Pharmazie - March 22, 2018 Category: Drugs & Pharmacology Source Type: research
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Archiv der Pharmazie, Ahead of Print. (Source: Archiv der Pharmazie)
Source: Archiv der Pharmazie - March 22, 2018 Category: Drugs & Pharmacology Source Type: research
Fungal biofilm inhibition by piperazine ‐sulphonamide linked Schiff bases: Design, synthesis, and biological evaluation
Archiv der Pharmazie, EarlyView. (Source: Archiv der Pharmazie)
Source: Archiv der Pharmazie - March 15, 2018 Category: Drugs & Pharmacology Source Type: research
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Archiv der Pharmazie, Ahead of Print. (Source: Archiv der Pharmazie)
Source: Archiv der Pharmazie - March 15, 2018 Category: Drugs & Pharmacology Source Type: research
Retracted: Novel spiro ‐thiazolidin‐4‐one and thioether derivatives of benzylidene flavanones: New leads in cancer and microbial chemotherapy
Archiv der Pharmazie, EarlyView. (Source: Archiv der Pharmazie)
Source: Archiv der Pharmazie - March 12, 2018 Category: Drugs & Pharmacology Authors: Sayeed Mukhtar
,
Meshari A. Alsharif
,
Mohammed I. Alahmdi
,
Humaira Parveen
,
Asad U. Khan Source Type: research
Synthesis, biological evaluation, and docking studies of some 5 ‐chloro‐2(3H)‐benzoxazolone Mannich bases derivatives as cholinesterase inhibitors
Archiv der Pharmazie, EarlyView. (Source: Archiv der Pharmazie)
Source: Archiv der Pharmazie - March 12, 2018 Category: Drugs & Pharmacology Source Type: research
Novel spiro ‐thiazolidin‐4‐one and thioether derivatives of benzylidene flavanones: New leads in cancer and microbial chemotherapy
Archiv der Pharmazie, EarlyView. (Source: Archiv der Pharmazie)
Source: Archiv der Pharmazie - March 12, 2018 Category: Drugs & Pharmacology Source Type: research
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Archiv der Pharmazie, Ahead of Print. (Source: Archiv der Pharmazie)
Source: Archiv der Pharmazie - March 12, 2018 Category: Drugs & Pharmacology Source Type: research
Synthesis, biological evaluation, and docking studies of some 5 ‐chloro‐2(3H)‐benzoxazolone Mannich bases derivatives as cholinesterase inhibitors
Abstract
A series of N‐substituted‐5‐chloro‐2(3H)‐benzoxazolone derivatives were synthesized and evaluated for their acetylcholinesterase (AChE), butyrylcholinesterase (BuChE) inhibitory, and antioxidant activities. The structures of the title compounds were confirmed by spectral and elemental analyses. The cholinesterase (ChE) inhibitory activity studies were carried out using Ellman's colorimetric method. The free radical scavenging activity was also determined by in vitro ABTS (2,2‐azinobis(3‐ethylbenzothiazoline‐6‐sulfonic acid)) assay. The biological activity results revealed that all of the title co...
Source: Archiv der Pharmazie - March 12, 2018 Category: Drugs & Pharmacology Authors: Sirin Uysal, Sulunay Parlar, Ayse H. Tarikogullari, Fadime Aydin Kose, Vildan Alptuzun, Zeynep Soyer Tags: FULL PAPER Source Type: research
Non ‐peptide‐based new class of platelet aggregation inhibitors: Design, synthesis, bioevaluation, SAR, and in silico studies
Archiv der Pharmazie, EarlyView. (Source: Archiv der Pharmazie)
Source: Archiv der Pharmazie - March 9, 2018 Category: Drugs & Pharmacology Source Type: research
Pyridine ‐substituted thiazolylphenol derivatives: Synthesis, modeling studies, aromatase inhibition, and antiproliferative activity evaluation
Archiv der Pharmazie, EarlyView. (Source: Archiv der Pharmazie)
Source: Archiv der Pharmazie - March 9, 2018 Category: Drugs & Pharmacology Source Type: research
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Archiv der Pharmazie, Ahead of Print. (Source: Archiv der Pharmazie)
Source: Archiv der Pharmazie - March 9, 2018 Category: Drugs & Pharmacology Source Type: research
