Recent advancements in DVD-Ig based therapeutic development
Publication date: Available online 20 November 2020Source: Drug Discovery Today: TechnologiesAuthor(s): Feng Dong, Tariq Ghayur (Source: Drug Discovery Today: Technologies)
Source: Drug Discovery Today: Technologies - November 21, 2020 Category: Drugs & Pharmacology Source Type: research

Graph-based generative models for de Novo drug design
Publication date: Available online 21 November 2020Source: Drug Discovery Today: TechnologiesAuthor(s): Xiaolin Xia, Jianxing Hu, Yanxing Wang, Liangren Zhang, Zhenming Liu (Source: Drug Discovery Today: Technologies)
Source: Drug Discovery Today: Technologies - November 21, 2020 Category: Drugs & Pharmacology Source Type: research

Synthetic carbohydrate-based HIV-1 vaccines
Publication date: Available online 29 October 2020Source: Drug Discovery Today: TechnologiesAuthor(s): Iñaki Bastida, Alberto Fernández-Tejada (Source: Drug Discovery Today: Technologies)
Source: Drug Discovery Today: Technologies - October 30, 2020 Category: Drugs & Pharmacology Source Type: research

Broadly protective semi-synthetic glycoconjugate vaccine against pathogens capable of producing poly-β-(1→6)-N-acetyl-d-glucosamine exopolysaccharide
Publication date: Available online 26 October 2020Source: Drug Discovery Today: TechnologiesAuthor(s): Marina L. Gening, Gerald B. Pier, Nikolay E. Nifantiev (Source: Drug Discovery Today: Technologies)
Source: Drug Discovery Today: Technologies - October 27, 2020 Category: Drugs & Pharmacology Source Type: research

On failure modes in molecule generation and optimization
Publication date: Available online 24 October 2020Source: Drug Discovery Today: TechnologiesAuthor(s): Philipp Renz, Dries Van Rompaey, Jörg Kurt Wegner, Sepp Hochreiter, Günter Klambauer (Source: Drug Discovery Today: Technologies)
Source: Drug Discovery Today: Technologies - October 24, 2020 Category: Drugs & Pharmacology Source Type: research

Viral safety for biotherapeutics and biosimilar
Publication date: Available online 14 October 2020Source: Drug Discovery Today: TechnologiesAuthor(s): Horst Ruppach (Source: Drug Discovery Today: Technologies)
Source: Drug Discovery Today: Technologies - October 14, 2020 Category: Drugs & Pharmacology Source Type: research

Bacterial polysaccharides: conformation, dynamics and molecular recognition by antibodies
Publication date: Available online 11 October 2020Source: Drug Discovery Today: TechnologiesAuthor(s): Marcos Gómez-Redondo, Ana Ardá, Ana Gimeno, Jesús Jiménez-Barbero (Source: Drug Discovery Today: Technologies)
Source: Drug Discovery Today: Technologies - October 12, 2020 Category: Drugs & Pharmacology Source Type: research

Carbohydrate-based adjuvants
Publication date: Available online 9 October 2020Source: Drug Discovery Today: TechnologiesAuthor(s): Pilar Garcia-Vello, Immacolata Speciale, Fabrizio Chiodo, Antonio Molinaro, Cristina De Castro (Source: Drug Discovery Today: Technologies)
Source: Drug Discovery Today: Technologies - October 9, 2020 Category: Drugs & Pharmacology Source Type: research

Efficient molecular encoders for virtual screening
Publication date: Available online 4 October 2020Source: Drug Discovery Today: TechnologiesAuthor(s): Youjun Xu, Chenjing Cai, Shiwei Wang, Luhua Lai, Jianfeng Pei (Source: Drug Discovery Today: Technologies)
Source: Drug Discovery Today: Technologies - October 4, 2020 Category: Drugs & Pharmacology Source Type: research

Antibody-drug conjugates as targeted therapies: Are we there yet? A critical review of the current clinical landscape
Publication date: Available online 29 September 2020Source: Drug Discovery Today: TechnologiesAuthor(s): Edit Tarcsa, Magali R. Guffroy, Hadi Falahatpisheh, Colin Phipps, John C. Kalvass (Source: Drug Discovery Today: Technologies)
Source: Drug Discovery Today: Technologies - September 29, 2020 Category: Drugs & Pharmacology Source Type: research

Selecting machine-learning scoring functions for structure-based virtual screening
Publication date: Available online 19 September 2020Source: Drug Discovery Today: TechnologiesAuthor(s): Pedro J. Ballester (Source: Drug Discovery Today: Technologies)
Source: Drug Discovery Today: Technologies - September 20, 2020 Category: Drugs & Pharmacology Source Type: research

Proteochemometrics – recent developments in bioactivity and selectivity modeling
Publication date: Available online 20 September 2020Source: Drug Discovery Today: TechnologiesAuthor(s): Brandon J. Bongers, Adriaan. P. IJzerman, Gerard J.P. Van Westen (Source: Drug Discovery Today: Technologies)
Source: Drug Discovery Today: Technologies - September 20, 2020 Category: Drugs & Pharmacology Source Type: research

Current methods and challenges for deep learning in drug discovery
Publication date: Available online 17 August 2020Source: Drug Discovery Today: TechnologiesAuthor(s): Stefan Schroedl (Source: Drug Discovery Today: Technologies)
Source: Drug Discovery Today: Technologies - August 18, 2020 Category: Drugs & Pharmacology Source Type: research

The good, the bad, and the ugly in chemical and biological data for machine learning
Publication date: Available online 26 July 2020Source: Drug Discovery Today: TechnologiesAuthor(s): Tiago Rodrigues (Source: Drug Discovery Today: Technologies)
Source: Drug Discovery Today: Technologies - July 26, 2020 Category: Drugs & Pharmacology Source Type: research

Practical considerations for active machine learning in drug discovery
Publication date: Available online 19 July 2020Source: Drug Discovery Today: TechnologiesAuthor(s): Daniel Reker (Source: Drug Discovery Today: Technologies)
Source: Drug Discovery Today: Technologies - July 20, 2020 Category: Drugs & Pharmacology Source Type: research