Escape from planarity in fragment-based drug discovery: A physicochemical and 3D property analysis of synthetic 3D fragment libraries

Publication date: Available online 17 June 2021Source: Drug Discovery Today: TechnologiesAuthor(s): David J. Hamilton, Tom Dekker, Hanna F. Klein, Guido V. Janssen, Maikel Wijtmans, Peter O’Brien, Iwan J.P. de Esch
Source: Drug Discovery Today: Technologies - Category: Drugs & Pharmacology Source Type: research