An iminium ion metabolite hampers the production of the pharmacologically active metabolite of a multikinase inhibitor KW ‐2449 in primates: irreversible inhibition of aldehyde oxidase and covalent binding with endogenous proteins

Biopharmaceutics&Drug Disposition,Volume 39, Issue 3, Page 164-174, March 2018.
Source: Biopharmaceutics and Drug Disposition - Category: Drugs & Pharmacology Source Type: research