Etravirine

Etravirine, also known as Intelence or TMC125, is a diarylpyrimidine (DAPY) derivative with potent in vitro activity against HIV. [#] In vitro, etravirine has equipotent activity against wild-type HIV and NNRTI-resistant variants that encode L100I, K103N, Y181C, Y188L, and G190A/S mutations. [#]
Source: Aids Info Drugs - Category: Drugs & Pharmacology Source Type: research